The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor
2017-01-01 Wapenaar, H; van den Bosch, T; Leus, Ngj; van der Wouden, Pe; Eleftheriadis, N; Hermans, J; Hailu, Gs; Rotili, D; Mai, A; Dömling, A; Bischoff, R; Haisma, Hj; Dekker, F. J.
A novel orally active water-soluble inhibitor of human glutathione transferase exerts a potent and selective antitumor activity against human melanoma xenografts
2015-01-01 De Luca, Anastasia; Rotili, Dante; Carpanese, Debora; Lenoci, Alessia; Calderan, Laura; Scimeca, Manuel; Mai, Antonello; Bonanno, Elena; Rosato, Antonio; Geroni, Cristina; Quintieri, Luigi; Caccuri, Anna Maria
Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural features
2016-01-01 Speranzini, Valentina; Rotili, Dante; Ciossani, Giuseppe; Pilotto, Simona; Marrocco, Biagina; Forgione, Mariantonietta; Lucidi, Alessia; Forneris, Federico; Mehdipour, Parinaz; Velankar, Sameer; Mai, Antonello; Mattevi, Andrea
Characterization of Sirtuin Inhibitors in Nematodes Expressing a Muscular Dystrophy Protein Reveals Muscle Cell and Behavioral Protection by Specific Sirtinol Analogues
2010-01-01 Matthieu Y., Pasco; Rotili, Dante; Lucia, Altucci; Francesca, Farina; Guy A., Rouleau; Mai, Antonello; Christian, Neri
Lysine deacetylase inhibitors in parasites: past, present, and future perspectives
2017-01-01 Hailu, Gs; Robaa, D; Forgione, M; Sippl, W; Rotili, D; Mai, A.
Selective class II HDAC inhibitors impair myogenesis by modulating the stability and activity of HDAC-MEF2 complexes
2009-01-01 Nebbioso, A; Manzo, F; Miceli, M; Conte, M; Manente, L; Baldi, A; De Luca, A; Rotili, Dante; Valente, Sergio; Mai, Antonello; Usiello, A; Gronemeyer, H; Altucci, L.
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases
2009-01-01 Mai, Antonello; Rotili, Dante; Tarantino, Domenico; Angela, Nebbioso; Sabrina, Castellano; Gianluca, Sbardella; Marc, Tini; Lucia, Altucci
Inhibition of histone demethylases LSD1 and UTX regulates ERα signaling in breast cancer
2019-01-01 Benedetti, R.; Dell'Aversana, C.; De Marchi, T.; Rotili, D.; Liu, N. Q.; Novakovic, B.; Boccella, S.; Di Maro, S.; Cosconati, S.; Baldi, A.; Nimeus, E.; Schultz, J.; Hoglund, U.; Maione, S.; Papulino, C.; Chianese, U.; Iovino, F.; Federico, A.; Mai, A.; Stunnenberg, H. G.; Nebbioso, A.; Altucci, L.
Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cells
2014-01-01 Lenoci, Alessia; Tomassi, S; Conte, M; Benedetti, R; Rodriguez, V; Carradori, Simone; Secci, Daniela; Castellano, S; Sbardella, G; Filetici, P; Novellino, E; Altucci, L; Rotili, Dante; Mai, Antonello
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties
2006-01-01 A, Mai; Rotili, D.; D, Tarantino; P, Ornaghi; F, Tosi; C, Vicidomini; G, Sbardella; A, Nebbioso; M, Miceli; L, Altucci; P, Filetici
The histone deacetylase inhibitor suberoylanilide hydroxamic acid reduces cardiac arrhythmias in dystrophic mice
2010-01-01 C., Colussi; R., Berni; J., Rosati; S., Straino; S., Vitale; F., Spallotta; S., Baruffi; L., Bocchi; F., Delucchi; S., Rossi; M., Savi; Rotili, Dante; F., Quaini; E., Macchi; D., Stilli; E., Musso; Mai, Antonello; Gaetano C., Capogrossi Mc
Sirtuin modulators: past, present, and future perspectives
2022-01-01 Fiorentino, Francesco; Mautone, Nicola; Menna, Martina; D'Acunzo, Francesca; Mai, Antonello; Rotili, Dante
Analytical and semipreparative high performance liquid chromatography separation of stereoisomers of novel 3,4-dihydropyrimidin-4(3H)-one derivatives on the immobilised amylose-based Chiralpack IA chiral stationary phase
2006-01-01 Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Mai, Antonello; Rotili, Dante
Chiral HPLC separation and absolute configuration of novel S-DABO derivatives
2009-01-01 Cirilli, R; Ferretti, R; LA TORRE, F; Borioni, A; Fares, V; Camalli, M; Faggi, C; Rotili, Dante; Mai, Antonello
A Photoreactive Small-Molecule Probe for 2-Oxoglutarate Oxygenases
2011-01-01 Rotili, Dante; Mikael, Altun; Akane, Kawamura; Alexander, Wolf; Roman, Fischer; I. k., Leung; Mukram m, Mackeen; Ya Min, Tian; Peter j, Ratcliffe; Mai, Antonello; Benedikt m, Kessler; Christopher j, Schofield
Histone deacetylase inhibitors and neurodegenerative disorders: Holding the promise
2009-01-01 Mai, Antonello; Rotili, Dante; Valente, Sergio; Aleksey, Kazantsev
Novel uracil-based 2-aminoanilide and 2-aminoanilide-like derivatives: Histone deacetylase inhibition and in-cell activities
2008-01-01 Mai, Antonello; Andrea, Perrone; Angela, Nebbioso; Rotili, Dante; Valente, Sergio; Maria, Tardugno; Silvio, Massa; Floriana De, Bellis; Lucia, Altucci
A new water soluble MAPK activator exerts antitumor activity in melanoma cells resistant to the BRAF inhibitor vemurafenib
2015-01-01 Graziani, Grazia; Artuso, Simona; De Luca, Anastasia; Muzi, Alessia; Rotili, Dante; Scimeca, Manuel; Atzori, Maria Grazia; Ceci, Claudia; Mai, Antonello; Leonetti, Carlo; Levati, Lauretta; Bonanno, Elena; Tentori, Lucio; Caccuri, Anna Maria
SIRT5 regulation of ammonia-induced autophagy and mitophagy
2015-01-01 Polletta, Lucia; Vernucci, Enza; Carnevale, Ilaria; Arcangeli, Tania; Rotili, Dante; Palmerio, Silvia; Steegborn, Clemens; Nowak, Theresa; Schutkowski, Mike; Pellegrini, Laura; Sansone, Luigi; Villanova, Lidia; Runci, Alessandra; Pucci, Bruna; Morgante, Emanuela; Fini, Massimo; Mai, Antonello; Russo, Matteo A; Tafani, Marco
Novel histone deacetylase inhibitors induce growth arrest, apoptosis, and differentiation in sarcoma cancer stem cells
2015-01-01 G., Di Pompo; M., Salerno; Rotili, Dante; Valente, Sergio; Zwergel, Clemens; S., Avnet; G., Lattanzi; N., Baldini; Mai, Antonello
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor | 1-gen-2017 | Wapenaar, H; van den Bosch, T; Leus, Ngj; van der Wouden, Pe; Eleftheriadis, N; Hermans, J; Hailu, Gs; Rotili, D; Mai, A; Dömling, A; Bischoff, R; Haisma, Hj; Dekker, F. J. | |
| A novel orally active water-soluble inhibitor of human glutathione transferase exerts a potent and selective antitumor activity against human melanoma xenografts | 1-gen-2015 | De Luca, Anastasia; Rotili, Dante; Carpanese, Debora; Lenoci, Alessia; Calderan, Laura; Scimeca, Manuel; Mai, Antonello; Bonanno, Elena; Rosato, Antonio; Geroni, Cristina; Quintieri, Luigi; Caccuri, Anna Maria | |
| Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural features | 1-gen-2016 | Speranzini, Valentina; Rotili, Dante; Ciossani, Giuseppe; Pilotto, Simona; Marrocco, Biagina; Forgione, Mariantonietta; Lucidi, Alessia; Forneris, Federico; Mehdipour, Parinaz; Velankar, Sameer; Mai, Antonello; Mattevi, Andrea | |
| Characterization of Sirtuin Inhibitors in Nematodes Expressing a Muscular Dystrophy Protein Reveals Muscle Cell and Behavioral Protection by Specific Sirtinol Analogues | 1-gen-2010 | Matthieu Y., Pasco; Rotili, Dante; Lucia, Altucci; Francesca, Farina; Guy A., Rouleau; Mai, Antonello; Christian, Neri | |
| Lysine deacetylase inhibitors in parasites: past, present, and future perspectives | 1-gen-2017 | Hailu, Gs; Robaa, D; Forgione, M; Sippl, W; Rotili, D; Mai, A. | |
| Selective class II HDAC inhibitors impair myogenesis by modulating the stability and activity of HDAC-MEF2 complexes | 1-gen-2009 | Nebbioso, A; Manzo, F; Miceli, M; Conte, M; Manente, L; Baldi, A; De Luca, A; Rotili, Dante; Valente, Sergio; Mai, Antonello; Usiello, A; Gronemeyer, H; Altucci, L. | |
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases | 1-gen-2009 | Mai, Antonello; Rotili, Dante; Tarantino, Domenico; Angela, Nebbioso; Sabrina, Castellano; Gianluca, Sbardella; Marc, Tini; Lucia, Altucci | |
| Inhibition of histone demethylases LSD1 and UTX regulates ERα signaling in breast cancer | 1-gen-2019 | Benedetti, R.; Dell'Aversana, C.; De Marchi, T.; Rotili, D.; Liu, N. Q.; Novakovic, B.; Boccella, S.; Di Maro, S.; Cosconati, S.; Baldi, A.; Nimeus, E.; Schultz, J.; Hoglund, U.; Maione, S.; Papulino, C.; Chianese, U.; Iovino, F.; Federico, A.; Mai, A.; Stunnenberg, H. G.; Nebbioso, A.; Altucci, L. | |
| Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cells | 1-gen-2014 | Lenoci, Alessia; Tomassi, S; Conte, M; Benedetti, R; Rodriguez, V; Carradori, Simone; Secci, Daniela; Castellano, S; Sbardella, G; Filetici, P; Novellino, E; Altucci, L; Rotili, Dante; Mai, Antonello | |
| Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties | 1-gen-2006 | A, Mai; Rotili, D.; D, Tarantino; P, Ornaghi; F, Tosi; C, Vicidomini; G, Sbardella; A, Nebbioso; M, Miceli; L, Altucci; P, Filetici | |
| The histone deacetylase inhibitor suberoylanilide hydroxamic acid reduces cardiac arrhythmias in dystrophic mice | 1-gen-2010 | C., Colussi; R., Berni; J., Rosati; S., Straino; S., Vitale; F., Spallotta; S., Baruffi; L., Bocchi; F., Delucchi; S., Rossi; M., Savi; Rotili, Dante; F., Quaini; E., Macchi; D., Stilli; E., Musso; Mai, Antonello; Gaetano C., Capogrossi Mc | |
| Sirtuin modulators: past, present, and future perspectives | 1-gen-2022 | Fiorentino, Francesco; Mautone, Nicola; Menna, Martina; D'Acunzo, Francesca; Mai, Antonello; Rotili, Dante | |
| Analytical and semipreparative high performance liquid chromatography separation of stereoisomers of novel 3,4-dihydropyrimidin-4(3H)-one derivatives on the immobilised amylose-based Chiralpack IA chiral stationary phase | 1-gen-2006 | Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Mai, Antonello; Rotili, Dante | |
| Chiral HPLC separation and absolute configuration of novel S-DABO derivatives | 1-gen-2009 | Cirilli, R; Ferretti, R; LA TORRE, F; Borioni, A; Fares, V; Camalli, M; Faggi, C; Rotili, Dante; Mai, Antonello | |
| A Photoreactive Small-Molecule Probe for 2-Oxoglutarate Oxygenases | 1-gen-2011 | Rotili, Dante; Mikael, Altun; Akane, Kawamura; Alexander, Wolf; Roman, Fischer; I. k., Leung; Mukram m, Mackeen; Ya Min, Tian; Peter j, Ratcliffe; Mai, Antonello; Benedikt m, Kessler; Christopher j, Schofield | |
| Histone deacetylase inhibitors and neurodegenerative disorders: Holding the promise | 1-gen-2009 | Mai, Antonello; Rotili, Dante; Valente, Sergio; Aleksey, Kazantsev | |
| Novel uracil-based 2-aminoanilide and 2-aminoanilide-like derivatives: Histone deacetylase inhibition and in-cell activities | 1-gen-2008 | Mai, Antonello; Andrea, Perrone; Angela, Nebbioso; Rotili, Dante; Valente, Sergio; Maria, Tardugno; Silvio, Massa; Floriana De, Bellis; Lucia, Altucci | |
| A new water soluble MAPK activator exerts antitumor activity in melanoma cells resistant to the BRAF inhibitor vemurafenib | 1-gen-2015 | Graziani, Grazia; Artuso, Simona; De Luca, Anastasia; Muzi, Alessia; Rotili, Dante; Scimeca, Manuel; Atzori, Maria Grazia; Ceci, Claudia; Mai, Antonello; Leonetti, Carlo; Levati, Lauretta; Bonanno, Elena; Tentori, Lucio; Caccuri, Anna Maria | |
| SIRT5 regulation of ammonia-induced autophagy and mitophagy | 1-gen-2015 | Polletta, Lucia; Vernucci, Enza; Carnevale, Ilaria; Arcangeli, Tania; Rotili, Dante; Palmerio, Silvia; Steegborn, Clemens; Nowak, Theresa; Schutkowski, Mike; Pellegrini, Laura; Sansone, Luigi; Villanova, Lidia; Runci, Alessandra; Pucci, Bruna; Morgante, Emanuela; Fini, Massimo; Mai, Antonello; Russo, Matteo A; Tafani, Marco | |
| Novel histone deacetylase inhibitors induce growth arrest, apoptosis, and differentiation in sarcoma cancer stem cells | 1-gen-2015 | G., Di Pompo; M., Salerno; Rotili, Dante; Valente, Sergio; Zwergel, Clemens; S., Avnet; G., Lattanzi; N., Baldini; Mai, Antonello |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile
Scopri
Tipologia
- 1 Contributo su Rivista58567
- 4 Contributo in Atti di Convegno ...1
Data di pubblicazione
- In corso di stampa166
- 2020 - 202715137
- 2010 - 201920733
- 2000 - 200914183
- 1990 - 19995643
- 1980 - 19892064
- 1970 - 1979621
- 1966 - 196922
Editore
- Giappichelli2
- Springer2
- -Attuale :ELSEVIER SCIENCE BV, PO...1
- Aracne1
- Aracne Editrice1
- Associazione Idrotecnica italiana1
- Astronomical Society of the Pacific1
- Bollettino Società Italiana di Fi...1
- Compumag 20131
- Editorial Academia del Hispanismo1
Rivista
- PHYSICS LETTERS. SECTION B674
- JOURNAL OF HIGH ENERGY PHYSICS453
- PHYSICAL REVIEW LETTERS388
- ASTRONOMY & ASTROPHYSICS385
- THE EUROPEAN PHYSICAL JOURNAL. C,...376
- CADMO260
- PHYSICAL REVIEW D259
- FEDERALISMI.IT252
- MONTHLY NOTICES OF THE ROYAL ASTR...240
- PHYSICAL REVIEW D, PARTICLES, FIE...201
Serie
- ATTUALITÀ COSTITUZIONALE1
- L’UNITÀ DEL DIRITTO1
Keyword
- Italy277
- Humans237
- Nuclear and High Energy Physics193
- Roma151
- Electrical and Electronic Enginee...148
- Hadron-Hadron Scattering141
- Physics and Astronomy (miscellane...139
- Condensed Matter Physics135
- Male125
- Ecology121
Lingua
- eng28417
- ita20347
- fre638
- spa625
- ger200
- por126
- lat59
- und59
- rus42
- cat17
Accesso al fulltext
- no fulltext55695
- open2834
- restricted30
- partially open5
- reserved4
- embargoed1