Pharmacological targeting of CBP/p300 drives a redox/autophagy axis leading to senescence-induced growth arrest in non-small cell lung cancer cells
2023-01-01 Ansari, Mohammad Salik Zeya; Stagni, Venturina; Iuzzolino, Angela; Rotili, Dante; Mai, Antonello; Del Bufalo, Donatella; Lavia, Patrizia; Degrassi, Francesca; Trisciuoglio, Daniela
The role of structural biology in the design of sirtuin activators
2023-01-01 Fiorentino, Francesco; Mai, Antonello; Rotili, Dante
Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells
2023-01-01 Zwergel, Clemens; Aventaggiato, Michele; Garbo, Sabrina; Di Bello, Elisabetta; Fassari, Bruno; Noce, Beatrice; Castiello, Carola; Lambona, Chiara; Barreca, Federica; Rotili, Dante; Fioravanti, Rossella; Schmalz, Thomas; Weyand, Michael; Niedermeier, Amelie; Tripodi, Marco; Colotti, Gianni; Steegborn, Clemens; Battistelli, Cecilia; Tafani, Marco; Valente, Sergio; Mai, Antonello
Emerging Roles of SIRT5 in Metabolism, Cancer, and SARS-CoV-2 Infection
2023-01-01 Fabbrizi, Emanuele; Fiorentino, Francesco; Carafa, Vincenzo; Altucci, Lucia; Mai, Antonello; Rotili, Dante
Role of SIRT3 in Microgravity Response: A New Player in Muscle Tissue Recovery
2023-01-01 Aventaggiato, Michele; Barreca, Federica; Vitiello, Laura; Vespa, Simone; Valente, Sergio; Rotili, Dante; Mai, Antonello; Lotti, Lavinia Vittoria; Sansone, Luigi; Russo, Matteo A.; Bizzarri, Mariano; Ferretti, Elisabetta; Tafani, Marco
Native mass spectrometry-directed drug discovery: Recent advances in investigating protein function and modulation
2023-01-01 Fiorentino, Francesco; Rotili, Dante; Mai, Antonello
Chemically Diverse S. mansoni HDAC8 Inhibitors Reduce Viability in Worm Larval and Adult Stages
2023-01-01 Noce, Beatrice; Di Bello, Elisabetta; Zwergel, Clemens; Fioravanti, Rossella; Valente, Sergio; Rotili, Dante; Masotti, Andrea; Salik Zeya Ansari, Mohammad; Trisciuoglio, Daniela; Chakrabarti, Alokta; Romier, Christophe; Robaa, Dina; Sippl, Wolfgang; Jung, Manfred; Häberli, Cécile; Keiser, Jennifer; Mai, Antonello
Modulation of Virulence-Associated Traits in Aspergillus fumigatus by BET Inhibitor JQ1
2022-01-01 Orekhova, Anastasia; De Angelis, Marta; Cacciotti, Andrea; Reverberi, Massimo; Rotili, Dante; Giorgi, Alessandra; Protto, Virginia; Bonincontro, Graziana; Fiorentino, Francesco; Zgoda, Victor; Mai, Antonello; Palamara, Anna Teresa; Simonetti, Giovanna
Neuroprotective Effects of PARP Inhibitors in Drosophila Models of Alzheimer’s Disease
2022-01-01 Maggiore, Anna; Casale, Assunta Maria; Toscanelli, Walter; Cappucci, Ugo; Rotili, Dante; Grieco, Maddalena; Gagné, Jean-Philippe; Poirier, Guy G.; D'Erme, Maria; Piacentini, Lucia
Biochemical Functions and Clinical Characterizations of the Sirtuins in Diabetes-Induced Retinal Pathologies
2022-01-01 Taurone, Samanta; De Ponte, Chiara; Rotili, Dante; De Santis, Elena; Mai, Antonello; Fiorentino, Francesco; Scarpa, Susanna; Artico, Marco; Micera, Alessandra
The Nitrobenzoxadiazole Derivative NBDHEX Behaves as Plasmodium falciparum Gametocyte Selective Inhibitor with Malaria Parasite Transmission Blocking Activity
2022-01-01 Siciliano, Giulia; Di Paolo, Veronica; Rotili, Dante; Migale, Rossella; Pedini, Francesca; Casella, Marialuisa; Camerini, Serena; Dalzoppo, Daniele; Henderson, Rob; Huijs, Tonnie; Dechering, Koen J.; Mai, Antonello; Caccuri, Anna Maria; Lalle, Marco; Quintieri, Luigi; Alano, Pietro
A potent HDAC inhibitor blocks Toxoplasma gondii tachyzoite growth and profoundly disrupts parasite gene expression
2022-01-01 Mouveaux, Thomas; Rotili, Dante; Boissavy, Tom; Roger, Emmanuel; Pierrot, Christine; Mai, Antonello; Gissot, Mathieu
Multimodal evaluation of 19F-BPA internalization in pancreatic cancer cells for boron capture and proton therapy potential applications
2022-01-01 Ciardiello, Andrea; Altieri, Saverio; Ballarini, Francesca; Bocci, Valerio; Bortolussi, Silva; Cansolino, Laura; Carlotti, Daniele; Ciocca, Mario; Faccini, Riccardo; Facoetti, Angelica; Ferrari, Cinzia; Ficcadenti, Luca; Furfaro, Emiliano; Giagu, Stefano; Iacoangeli, Francesco; Macioce, Giampiero; Mancini-Terracciano, Carlo; Messina, Andrea; Milazzo, Luisa; Pacifico, Severina; Piccolella, Simona; Postuma, Ian; Rotili, Dante; Vercesi, Valerio; Voena, Cecilia; Vulcano, Francesca; Capuani, Silvia
Mass spectrometry enables the discovery of inhibitors of an LPS transport assembly via disruption of protein–protein interactions
2021-01-01 Fiorentino, Francesco; Rotili, Dante; Mai, Antonello; Bolla, Jani R.; Robinson, Carol V.
Anti-influenza A virus activity and structure–activity relationship of a series of nitrobenzoxadiazole derivatives
2021-01-01 Fiorentino, Francesco; De Angelis, Marta; Menna, Martina; Rovere, Annarita; Caccuri, Anna Maria; D'Acunzo, Francesca; Palamara, Anna Teresa; Nencioni, Lucia; Rotili, Dante; Mai, Antonello
SIRT5 Inhibition Induces Brown Fat-Like Phenotype in 3T3-L1 Preadipocytes
2021-01-01 Molinari, Francesca; Feraco, Alessandra; Mirabilii, Simone; Saladini, Serena; Sansone, Luigi; Vernucci, Enza; Tomaselli, Giada; Marzolla, Vincenzo; Rotili, Dante; Russo, Matteo A.; Ricciardi, Maria Rosaria; Tafuri, Agostino; Mai, Antonello; Caprio, Massimiliano; Tafani, Marco; Armani, Andrea
Regulatory Interplay between miR-181a-5p and Estrogen Receptor Signaling Cascade in Breast Cancer
2021-01-01 Benedetti, Rosaria; Papulino, Chiara; Sgueglia, Giulia; Chianese, Ugo; De Marchi, Tommaso; Iovino, Francesco; Rotili, Dante; Mai, Antonello; Niméus, Emma; Dell' Aversana, Carmela; Altucci, Lucia
Recent Advances in Epigenetic Proteolysis Targeting Chimeras (Epi-PROTACs)
2020-01-01 Tomaselli, Daniela; Mautone, Nicola; Mai, Antonello; Rotili, Dante
Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni
2020-01-01 Coutinho Carneiro, Vitor; De Abreu Da Silva, Isabel Caetano; Amaral, Murilo Sena; Pereira, Adriana S. A.; Silveira, Gilbert Oliveira; Pires, David Da Silva; Verjovski-Almeida, Sergio; Dekker, Frank J.; Rotili, Dante; Mai, Antonello; Lopes-Torres, Eduardo José; Robaa, Dina; Sippl, Wolfgang; Pierce, Raymond J.; Borrello, M. Teresa; Ganesan, A.; Lancelot, Julien; Thiengo, Silvana; Fernandez, Monica Ammon; Vicentino, Amanda Roberta Revoredo; Mourão, Marina Moraes; Coelho, Fernanda Sales; Fantappié, Marcelo Rosado
Identification of Inhibitors to Trypanosoma cruzi Sirtuins Based on Compounds Developed to Human Enzymes
2020-01-01 Matutino Bastos, Tanira; Botelho Pereira Soares, Milena; Haddad Franco, Caio; Alcântara, Laura; Antonini, Lorenzo; Sabatino, Manuela; Mautone, Nicola; Holanda Freitas-Junior, Lucio; Moraes, Carolina Borsoi; Ragno, Rino; Rotili, Dante; Schenkman, Sergio; Mai, Antonello; Silvio Moretti, Nilmar
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Pharmacological targeting of CBP/p300 drives a redox/autophagy axis leading to senescence-induced growth arrest in non-small cell lung cancer cells | 1-gen-2023 | Ansari, Mohammad Salik Zeya; Stagni, Venturina; Iuzzolino, Angela; Rotili, Dante; Mai, Antonello; Del Bufalo, Donatella; Lavia, Patrizia; Degrassi, Francesca; Trisciuoglio, Daniela | |
| The role of structural biology in the design of sirtuin activators | 1-gen-2023 | Fiorentino, Francesco; Mai, Antonello; Rotili, Dante | |
| Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells | 1-gen-2023 | Zwergel, Clemens; Aventaggiato, Michele; Garbo, Sabrina; Di Bello, Elisabetta; Fassari, Bruno; Noce, Beatrice; Castiello, Carola; Lambona, Chiara; Barreca, Federica; Rotili, Dante; Fioravanti, Rossella; Schmalz, Thomas; Weyand, Michael; Niedermeier, Amelie; Tripodi, Marco; Colotti, Gianni; Steegborn, Clemens; Battistelli, Cecilia; Tafani, Marco; Valente, Sergio; Mai, Antonello | |
| Emerging Roles of SIRT5 in Metabolism, Cancer, and SARS-CoV-2 Infection | 1-gen-2023 | Fabbrizi, Emanuele; Fiorentino, Francesco; Carafa, Vincenzo; Altucci, Lucia; Mai, Antonello; Rotili, Dante | |
| Role of SIRT3 in Microgravity Response: A New Player in Muscle Tissue Recovery | 1-gen-2023 | Aventaggiato, Michele; Barreca, Federica; Vitiello, Laura; Vespa, Simone; Valente, Sergio; Rotili, Dante; Mai, Antonello; Lotti, Lavinia Vittoria; Sansone, Luigi; Russo, Matteo A.; Bizzarri, Mariano; Ferretti, Elisabetta; Tafani, Marco | |
| Native mass spectrometry-directed drug discovery: Recent advances in investigating protein function and modulation | 1-gen-2023 | Fiorentino, Francesco; Rotili, Dante; Mai, Antonello | |
| Chemically Diverse S. mansoni HDAC8 Inhibitors Reduce Viability in Worm Larval and Adult Stages | 1-gen-2023 | Noce, Beatrice; Di Bello, Elisabetta; Zwergel, Clemens; Fioravanti, Rossella; Valente, Sergio; Rotili, Dante; Masotti, Andrea; Salik Zeya Ansari, Mohammad; Trisciuoglio, Daniela; Chakrabarti, Alokta; Romier, Christophe; Robaa, Dina; Sippl, Wolfgang; Jung, Manfred; Häberli, Cécile; Keiser, Jennifer; Mai, Antonello | |
| Modulation of Virulence-Associated Traits in Aspergillus fumigatus by BET Inhibitor JQ1 | 1-gen-2022 | Orekhova, Anastasia; De Angelis, Marta; Cacciotti, Andrea; Reverberi, Massimo; Rotili, Dante; Giorgi, Alessandra; Protto, Virginia; Bonincontro, Graziana; Fiorentino, Francesco; Zgoda, Victor; Mai, Antonello; Palamara, Anna Teresa; Simonetti, Giovanna | |
| Neuroprotective Effects of PARP Inhibitors in Drosophila Models of Alzheimer’s Disease | 1-gen-2022 | Maggiore, Anna; Casale, Assunta Maria; Toscanelli, Walter; Cappucci, Ugo; Rotili, Dante; Grieco, Maddalena; Gagné, Jean-Philippe; Poirier, Guy G.; D'Erme, Maria; Piacentini, Lucia | |
| Biochemical Functions and Clinical Characterizations of the Sirtuins in Diabetes-Induced Retinal Pathologies | 1-gen-2022 | Taurone, Samanta; De Ponte, Chiara; Rotili, Dante; De Santis, Elena; Mai, Antonello; Fiorentino, Francesco; Scarpa, Susanna; Artico, Marco; Micera, Alessandra | |
| The Nitrobenzoxadiazole Derivative NBDHEX Behaves as Plasmodium falciparum Gametocyte Selective Inhibitor with Malaria Parasite Transmission Blocking Activity | 1-gen-2022 | Siciliano, Giulia; Di Paolo, Veronica; Rotili, Dante; Migale, Rossella; Pedini, Francesca; Casella, Marialuisa; Camerini, Serena; Dalzoppo, Daniele; Henderson, Rob; Huijs, Tonnie; Dechering, Koen J.; Mai, Antonello; Caccuri, Anna Maria; Lalle, Marco; Quintieri, Luigi; Alano, Pietro | |
| A potent HDAC inhibitor blocks Toxoplasma gondii tachyzoite growth and profoundly disrupts parasite gene expression | 1-gen-2022 | Mouveaux, Thomas; Rotili, Dante; Boissavy, Tom; Roger, Emmanuel; Pierrot, Christine; Mai, Antonello; Gissot, Mathieu | |
| Multimodal evaluation of 19F-BPA internalization in pancreatic cancer cells for boron capture and proton therapy potential applications | 1-gen-2022 | Ciardiello, Andrea; Altieri, Saverio; Ballarini, Francesca; Bocci, Valerio; Bortolussi, Silva; Cansolino, Laura; Carlotti, Daniele; Ciocca, Mario; Faccini, Riccardo; Facoetti, Angelica; Ferrari, Cinzia; Ficcadenti, Luca; Furfaro, Emiliano; Giagu, Stefano; Iacoangeli, Francesco; Macioce, Giampiero; Mancini-Terracciano, Carlo; Messina, Andrea; Milazzo, Luisa; Pacifico, Severina; Piccolella, Simona; Postuma, Ian; Rotili, Dante; Vercesi, Valerio; Voena, Cecilia; Vulcano, Francesca; Capuani, Silvia | |
| Mass spectrometry enables the discovery of inhibitors of an LPS transport assembly via disruption of protein–protein interactions | 1-gen-2021 | Fiorentino, Francesco; Rotili, Dante; Mai, Antonello; Bolla, Jani R.; Robinson, Carol V. | |
| Anti-influenza A virus activity and structure–activity relationship of a series of nitrobenzoxadiazole derivatives | 1-gen-2021 | Fiorentino, Francesco; De Angelis, Marta; Menna, Martina; Rovere, Annarita; Caccuri, Anna Maria; D'Acunzo, Francesca; Palamara, Anna Teresa; Nencioni, Lucia; Rotili, Dante; Mai, Antonello | |
| SIRT5 Inhibition Induces Brown Fat-Like Phenotype in 3T3-L1 Preadipocytes | 1-gen-2021 | Molinari, Francesca; Feraco, Alessandra; Mirabilii, Simone; Saladini, Serena; Sansone, Luigi; Vernucci, Enza; Tomaselli, Giada; Marzolla, Vincenzo; Rotili, Dante; Russo, Matteo A.; Ricciardi, Maria Rosaria; Tafuri, Agostino; Mai, Antonello; Caprio, Massimiliano; Tafani, Marco; Armani, Andrea | |
| Regulatory Interplay between miR-181a-5p and Estrogen Receptor Signaling Cascade in Breast Cancer | 1-gen-2021 | Benedetti, Rosaria; Papulino, Chiara; Sgueglia, Giulia; Chianese, Ugo; De Marchi, Tommaso; Iovino, Francesco; Rotili, Dante; Mai, Antonello; Niméus, Emma; Dell' Aversana, Carmela; Altucci, Lucia | |
| Recent Advances in Epigenetic Proteolysis Targeting Chimeras (Epi-PROTACs) | 1-gen-2020 | Tomaselli, Daniela; Mautone, Nicola; Mai, Antonello; Rotili, Dante | |
| Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni | 1-gen-2020 | Coutinho Carneiro, Vitor; De Abreu Da Silva, Isabel Caetano; Amaral, Murilo Sena; Pereira, Adriana S. A.; Silveira, Gilbert Oliveira; Pires, David Da Silva; Verjovski-Almeida, Sergio; Dekker, Frank J.; Rotili, Dante; Mai, Antonello; Lopes-Torres, Eduardo José; Robaa, Dina; Sippl, Wolfgang; Pierce, Raymond J.; Borrello, M. Teresa; Ganesan, A.; Lancelot, Julien; Thiengo, Silvana; Fernandez, Monica Ammon; Vicentino, Amanda Roberta Revoredo; Mourão, Marina Moraes; Coelho, Fernanda Sales; Fantappié, Marcelo Rosado | |
| Identification of Inhibitors to Trypanosoma cruzi Sirtuins Based on Compounds Developed to Human Enzymes | 1-gen-2020 | Matutino Bastos, Tanira; Botelho Pereira Soares, Milena; Haddad Franco, Caio; Alcântara, Laura; Antonini, Lorenzo; Sabatino, Manuela; Mautone, Nicola; Holanda Freitas-Junior, Lucio; Moraes, Carolina Borsoi; Ragno, Rino; Rotili, Dante; Schenkman, Sergio; Mai, Antonello; Silvio Moretti, Nilmar |
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